Chemistry:Deschloroetizolam

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Short description: Chemical compound
Deschloroetizolam
Deschloroetizolam.svg
Deschloroetizolam.png
Clinical data
Dependence
liability
Moderate
Routes of
administration
Oral, sublingual, rectal
Legal status
Legal status
Identifiers
CAS Number
PubChem CID
ChemSpider
UNII
Chemical and physical data
FormulaC17H16N4S
Molar mass308.40 g·mol−1
3D model (JSmol)

Deschloroetizolam (also known as Etizolam-2) is a thienotriazolodiazepine that is the dechlorinated analog of the closely related etizolam.[1][2][3] The compound has been sold as a designer drug.[4][5][6][7]

Legal status

Deschloroetizolam is classified and controlled as a hazardous substance in Sweden as of on October 15, 2015.[8]

See also

References

  1. "Heteroaromaten mit anellierten Siebenringen, III. Umwandlung von Thienotriazolooxazepinen in Diazepine" (in German). Justus Liebigs Annalen der Chemie 1978 (8): 1257–1265. September 1978. doi:10.1002/jlac.197819780806. 
  2. Nakanishi M, Tahara T, Araki K, Shiroki M, "Triazolothienodiazepine compounds", US patent 3904641, published 1975-09-09, assigned to Yoshitomi Pharmaceutical Industries, Ltd.
  3. Hiroshi K, Syuji E, Hideaki S, Minoru M, Kenichi O, "Thienylazole compound and thienotriazolodiazepine compound", EP patent 0776892, published 4 June 1997, assigned to Yoshitomi Pharmaceutical Industries, Ltd.
  4. "Deschloroetizolam". New Synthetic Drugs Database. 9 November 2023. http://nsddb.eu/substance/374/. 
  5. "Detectability of designer benzodiazepines in CEDIA, EMIT II Plus, HEIA, and KIMS II immunochemical screening assays". Drug Testing and Analysis 9 (4): 640–645. April 2017. doi:10.1002/dta.2003. PMID 27366870. 
  6. "Experimental versus theoretical log D7.4 , pKa and plasma protein binding values for benzodiazepines appearing as new psychoactive substances". Drug Testing and Analysis 10 (8): 1258–1269. March 2018. doi:10.1002/dta.2387. PMID 29582576. https://rke.abertay.ac.uk/en/publications/527a634d-decc-4d3a-bdca-08659bb13ed6. 
  7. "The blood-to-plasma ratio and predicted GABAA-binding affinity of designer benzodiazepines". Forensic Toxicology 40 (2): 349–356. July 2022. doi:10.1007/s11419-022-00616-y. PMID 36454409. 
  8. "Nya substanser klassas som narkotika eller hälsofarlig vara" (in Swedish). Folkhälsomyndigheten. 18 August 2015. https://www.folkhalsomyndigheten.se/nyheter-och-press/nyhetsarkiv/2015/augusti/nya-substanser-klassas-som-narkotika-eller-halsofarlig-vara/.