Chemistry:Divaplon

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Short description: Chemical compound
Divaplon
Divaplon Structure.svg
Clinical data
ATC code
  • none
Identifiers
CAS Number
PubChem CID
ChemSpider
UNII
ChEMBL
Chemical and physical data
FormulaC17H17N3O2
Molar mass295.336 g·mol−1
3D model (JSmol)
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Divaplon (RU-32698) is a nonbenzodiazepine, anxiolytic and anticonvulsant drug from the imidazopyrimidine family of drugs. It acts as a partial agonist at the "benzodiazepine site" of the GABAA receptor in the brain.[1][2][3]

References

  1. "Lack of anticonvulsant tolerance with RU 32698 and Ro 17-1812". European Journal of Pharmacology 164 (2): 377–80. May 1989. doi:10.1016/0014-2999(89)90482-2. PMID 2759183. 
  2. "Benzodiazepine (omega) receptor partial agonists and the acquisition of conditioned fear in mice". Psychopharmacology 121 (1): 104–8. September 1995. doi:10.1007/BF02245596. PMID 8539334. 
  3. "Pharmacological analysis of the effects of benzodiazepines on punished schedule-induced polydipsia in rats". Behavioural Pharmacology 18 (1): 81–7. February 2007. doi:10.1097/FBP.0b013e3280143212. PMID 17218801.