Chemistry:CP-1414S

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Short description: Chemical compound
CP-1414S
CP-1414S.svg
Clinical data
ATC code
  • none
Identifiers
CAS Number
PubChem CID
ChemSpider
UNII
Chemical and physical data
FormulaC15H12N4O3
Molar mass296.286 g·mol−1
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CP-1414S is an experimental drug first made by a team in Germany.[1] It is a benzodiazepine derivative. CP-1414S is a 1,5-benzodiazepine, with the nitrogen atoms located at positions 1 and 5 of the diazepine ring, and so is most closely related to other 1,5-benzodiazepines such as clobazam.

CP-1414S has primarily anxiolytic and anticonvulsant effects.[2] Its potency is roughly equal to that of clobazam, but with more pronounced sedation.[3]

See also

References

  1. US Patent 3766169 PROCESS FOR THE PREPARATION OF 3-AMINOMETHYLIDENE-1,5-BENZODIAZEPINE-2,4-(3H,5H)-DIONES
  2. "Studies on some pharmacological activities of 7-nitro-2-amino-5-phenyl-3H-1,5-benzodiazepine (CP 1414 S) in the rat. A comparison with diazepam". Arzneimittel-Forschung 31 (10): 1721–3. 1981. PMID 6119091. 
  3. "Benzodiazepine receptors': correlation with pharmacological responses in living animals". Life Sciences 31 (19): 2025–35. November 1982. doi:10.1016/0024-3205(82)90094-7. PMID 6129557.